[A]
- Classes: All alpha proteins
- Folds: Bromodomain-like
- Superfamilies: alpha-ketoacid dehydrogenase kinase, N-terminal domain
- Families: alpha-ketoacid dehydrogenase kinase, N-terminal domain
- Protein Domains: automated matches
- Species: Human (Homo sapiens) [TaxId: 9606]
PDB Entries
PDB ID | OPM | Mutant | Chain Formula | Resolution | HETNAM | ||
---|---|---|---|---|---|---|---|
Amino Acid sequence | SCOPe Family Level | CATH Homology Level | |||||
2btz | [A2] | [A2] | [A2] | 2.2 | |||
2bu2 | [A2] | [A2] | [A2] | 2.4 | ATP:ADENOSINE-5___sq___-TRIPHOSPHATE MG:MAGNESIUM ION TF1:4-({(2R,5S)-2,5-DIMETHYL-4-[(2R)-3,3,3-TRIFLUORO-2-HYDROXY-2-METHYLPROPANOYL]PIPERAZIN-1-YL}CARBONYL)BENZONITRILE | ||
2bu5 | [A2] | [A2] | [A2] | 2.35 | TF1:4-({(2R,5S)-2,5-DIMETHYL-4-[(2R)-3,3,3-TRIFLUORO-2-HYDROXY-2-METHYLPROPANOYL]PIPERAZIN-1-YL}CARBONYL)BENZONITRILE | ||
2bu6 | [A2] | [A2] | [A2] | 2.4 | TF2:(N-{4-[(ETHYLANILINO)SULFONYL]-2-METHYLPHENYL}-3,3,3-TRIFLUORO-2-HYDROXY-2-METHYLPROPANAMIDE | ||
2bu7 | [A2] | [A2] | [A2] | 2.4 | TF3:N-(2-AMINOETHYL)-2-{3-CHLORO-4-[(4-ISOPROPYLBENZYL)OXY]PHENYL} ACETAMIDE | ||
2bu8 | [A2] | [A2] | [A2] | 2.5 | ADP:ADENOSINE-5___sq___-DIPHOSPHATE MG:MAGNESIUM ION TF4:DICHLORO-ACETIC ACID | ||
4mp2 | [A2] | [A2] | [A2] | 1.75 | PV1:(5-BROMO-2,4-DIHYDROXYPHENYL)(1,3-DIHYDRO-2H-ISOINDOL-2-YL)METHANONE TLA:L(+)-TARTARIC ACID | ||
4mp7 | [A2] | [A2] | [A2] | 1.8 | PFT:4-(1,3-DIHYDRO-2H-ISOINDOL-2-YLCARBONYL)BENZENE-1,3-DIOL TLA:L(+)-TARTARIC ACID | ||
4mpc | [A2] | [A2] | [A2] | 1.7 | PV2:4-(ISOINDOLIN-2-YLSULFONYL)BENZENE-1,3-DIOL TLA:L(+)-TARTARIC ACID | ||
4mpe | [A2] | [A2] | [A2] | 1.95 | PV8:4-[(5-HYDROXY-1,3-DIHYDRO-2H-ISOINDOL-2-YL)SULFONYL]BENZENE-1,3-DIOL TLA:L(+)-TARTARIC ACID | ||
4mpn | [A2] | [A2] | [A2] | 1.75 | PV0:2-[(2,4-DIHYDROXYPHENYL)SULFONYL]-2,3-DIHYDRO-1H-ISOINDOLE-4,6-DIOL TLA:L(+)-TARTARIC ACID | ||
4v25 | [A2] | [A2] | [A2] | 2.6 | MG:MAGNESIUM ION SZ6:N-[4-(2-CHLORO-5-METHYLPYRIMIDIN-4-YL)PHENYL]-N-(4-{[(DIFLUOROACETYL)AMINO]METHYL}BENZYL)-2,4-DIHYDROXYBENZAMIDE TF3:N-(2-AMINOETHYL)-2-{3-CHLORO-4-[(4-ISOPROPYLBENZYL)OXY]PHENYL} ACETAMIDE | ||
4v26 | [A2] | [A2] | [A2] | 2.49 | 7TJ:N-[4-(2-CHLORO-5-METHYLPYRIMIDIN-4-YL)PHENYL]-2,4-DIHYDROXY-N-(4-{[(TRIFLUOROACETYL)AMINO]METHYL}BENZYL)BENZAMIDE MG:MAGNESIUM ION TF3:N-(2-AMINOETHYL)-2-{3-CHLORO-4-[(4-ISOPROPYLBENZYL)OXY]PHENYL} ACETAMIDE | ||
5j6a | [A2] | [A2] | [A2] | 2.05 | P46:(3S)-3-AMINO-4-[4-({2-[(2,4-DIHYDROXYPHENYL)SULFONYL]-2H-ISOINDOL-5-YL}AMINO)PIPERIDIN-1-YL]-4-OXOBUTANAMIDE | ||
5j71 | [A2] | [A2] | [A2] | 1.65 | P35:4-({5-[(PIPERIDIN-4-YL)AMINO]-1,3-DIHYDRO-2H-ISOINDOL-2-YL}SULFONYL)BENZENE-1,3-DIOL TLA:L(+)-TARTARIC ACID | ||
5m4k | [A] | [A] | [A] | 2.6 | 7F9:~{N}-[2-(ETHYLAMINO)-2-OXIDANYLIDENE-ETHYL]-~{N}-(4-METHOXYPHENYL)-2,4-BIS(OXIDANYL)BENZAMIDE MG:MAGNESIUM ION TF3:N-(2-AMINOETHYL)-2-{3-CHLORO-4-[(4-ISOPROPYLBENZYL)OXY]PHENYL} ACETAMIDE | ||
5m4m | [A] | [A] | [A] | 2.4 | 7FW:~{N}-[4-[METHYL(QUINOXALIN-6-YLMETHYL)CARBAMOYL]PHENYL]-2,4-BIS(OXIDANYL)-~{N}-(PHENYLMETHYL)BENZAMIDE CL:CHLORIDE ION TF3:N-(2-AMINOETHYL)-2-{3-CHLORO-4-[(4-ISOPROPYLBENZYL)OXY]PHENYL} ACETAMIDE | ||
5m4n | [A] | [A] | [A] | 2.6 | 7FV:[2,4-BIS(OXIDANYL)PHENYL]-[(2~{S})-2-METHYL-6-(3-METHYLQUINOLIN-2-YL)-3,4-DIHYDRO-2~{H}-QUINOLIN-1-YL]METHANONE CL:CHLORIDE ION TF3:N-(2-AMINOETHYL)-2-{3-CHLORO-4-[(4-ISOPROPYLBENZYL)OXY]PHENYL} ACETAMIDE | ||
5m4p | [A] | [A] | [A] | 2.3 | 7FE:~{N}-[4-(2-CHLORANYL-5-METHYL-PYRIMIDIN-4-YL)PHENYL]-2,4-BIS(OXIDANYL)-~{N}-[[4-(PYRROLIDIN-1-YLMETHYL)PHENYL]METHYL]BENZAMIDE CL:CHLORIDE ION TF3:N-(2-AMINOETHYL)-2-{3-CHLORO-4-[(4-ISOPROPYLBENZYL)OXY]PHENYL} ACETAMIDE | ||
6lil | [A2] | [A2] | [A2] | 1.93 | EGX:1-(1-PIPERIDIN-4-YLPYRAZOL-4-YL)ANTHRACENE-9,10-DIONE FLC:CITRATE ANION GOL:GLYCEROL PEG:DI(HYDROXYETHYL)ETHER SO4:SULFATE ION | ||
6lin | [A2] | [A2] | [A2] | 2.67 | EH0:4-[[[4-[3,5-BIS(FLUORANYL)-4-(4-OXIDANYL-4-OXIDANYLIDENE-BUTOXY)PHENYL]-5-[5-CHLORANYL-2,4-BIS(OXIDANYL)PHENYL]-1,2-OXAZOL-3-YL]CARBONYLAMINO]METHYL]BENZOIC ACID GOL:GLYCEROL PEG:DI(HYDROXYETHYL)ETHER SO4:SULFATE ION | ||
6lio | [A2] | [A2] | [A2] | 1.76 | EH3:4-[[[5-[5-CHLORANYL-2,4-BIS(OXIDANYL)PHENYL]-4-[4-(1-METHYLSULFONYLPIPERIDIN-4-YL)OXYPHENYL]-1,2-OXAZOL-3-YL]CARBONYLAMINO]METHYL]CYCLOHEXANE-1-CARBOXYLIC ACID GOL:GLYCEROL SO4:SULFATE ION |
*Chain Formula of OLIGAMI.
[ ] : Polypeptide - [AB] : Protein, [ab] : Small peptide
( ) : Nucleic acid - (AB) : DNA, (ab) : RNA
[ ] : Polypeptide - [AB] : Protein, [ab] : Small peptide
( ) : Nucleic acid - (AB) : DNA, (ab) : RNA