[A][a]
- Classes: All alpha proteins
- Folds: HD-domain/PDEase-like
- Superfamilies: HD-domain/PDEase-like
- Families: PDEase
- Protein Domains: automated matches
- Species: Human (Homo sapiens) [TaxId: 9606]
PDB Entries
PDB ID | OPM | Mutant | Chain Formula | Resolution | HETNAM | ||
---|---|---|---|---|---|---|---|
Amino Acid sequence | SCOPe Family Level | CATH Homology Level | |||||
2qyk | [A] | [A] | [A] | 2.1 | MG:MAGNESIUM ION NPV:4-[8-(3-NITROPHENYL)-1,7-NAPHTHYRIDIN-6-YL]BENZOICACID ZN:ZINC ION | ||
2qym | [A2] | [A2] | [A2] | 1.9 | MG:MAGNESIUM ION ZN:ZINC ION | ||
2yy2 | [A2] | [A2] | [A2] | 2.8 | IBM:3-ISOBUTYL-1-METHYLXANTHINE MG:MAGNESIUM ION ZN:ZINC ION | ||
3i8v | [A2] | [A2] | [A2] | 2.25 | 0MO:(4R)-4-(3-BUTOXY-4-METHOXYBENZYL)IMIDAZOLIDIN-2-ONE CO:COBALT (II) ION CSS:S-MERCAPTOCYSTEINE GOL:GLYCEROL MG:MAGNESIUM ION ZN:ZINC ION | ||
3jwq | [A] | [A] | [A] | 2.87 | MG:MAGNESIUM ION VIA:5-{2-ETHOXY-5-[(4-METHYLPIPERAZIN-1-YL)SULFONYL]PHENYL}-1-METHYL-3-PROPYL-1H,6H,7H-PYRAZOLO[4,3-D]PYRIMIDIN-7-ONE ZN:ZINC ION | ||
3jwr | [A][a] | [A][a] | [A][a] | 2.99 | IBM:3-ISOBUTYL-1-METHYLXANTHINE MG:MAGNESIUM ION ZN:ZINC ION | ||
3o0j | [A] | [A] | [A] | 1.95 | 3OJ:4-[(1-HYDROXY-1,3-DIHYDRO-2,1-BENZOXABOROL-5-YL)OXY]BENZENE-1,2-DICARBONITRILE EDO:1,2-ETHANEDIOL MG:MAGNESIUM ION ZN:ZINC ION | ||
3qi3 | [A2] | [A2] | [A2] | 2.3 | MG:MAGNESIUM ION PDB:1-(2-CHLOROPHENYL)-6-[(2R)-3,3,3-TRIFLUORO-2-METHYLPROPYL]-1,7-DIHYDRO-4H-PYRAZOLO[3,4-D]PYRIMIDIN-4-ONE ZN:ZINC ION | ||
3shy | [A] | [A] | [A] | 2.65 | 5FO:6-ETHYL-5-FLUORO-2-{5-[(4-METHYLPIPERAZIN-1-YL)SULFONYL]-2-PROPOXYPHENYL}PYRIMIDIN-4(3H)-ONE MG:MAGNESIUM ION ZN:ZINC ION | ||
3shz | [A] | [A] | [A] | 2.45 | 5CO:5-CHLORO-6-ETHYL-2-{5-[(4-METHYLPIPERAZIN-1-YL)SULFONYL]-2-PROPOXYPHENYL}PYRIMIDIN-4(3H)-ONE MG:MAGNESIUM ION ZN:ZINC ION | ||
3sie | [A] | [A] | [A] | 1.93 | 5BO:5-BROMO-6-ETHYL-2-{5-[(4-METHYLPIPERAZIN-1-YL)SULFONYL]-2-PROPOXYPHENYL}PYRIMIDIN-4(3H)-ONE | ||
3tvx | [A] | [A] | [A] | 2.84 | MG:MAGNESIUM ION PNX:3,7-DIMETHYL-1-(5-OXOHEXYL)-3,7-DIHYDRO-1H-PURINE-2,6-DIONE SO4:SULFATE ION ZN:ZINC ION | ||
4g2w | [A] | [A] | [A] | 2.28 | MG:MAGNESIUM ION NI0:5,6-DIETHYL-2-{5-[(4-METHYLPIPERAZIN-1-YL)SULFONYL]-2-PROPOXYPHENYL}PYRIMIDIN-4(3H)-ONE PEG:DI(HYDROXYETHYL)ETHER ZN:ZINC ION | ||
4g2y | [A] | [A] | [A] | 2.4 | MG:MAGNESIUM ION NI5:2-{5-[(4-METHYLPIPERAZIN-1-YL)SULFONYL]-2-PROPOXYPHENYL}-3,5,6,7-TETRAHYDRO-4H-CYCLOPENTA[D]PYRIMIDIN-4-ONE PEG:DI(HYDROXYETHYL)ETHER ZN:ZINC ION | ||
4i9z | [A] | [A] | [A] | 2.08 | 5BA:5-BROMO-2-{5-[(4-METHYLPIPERAZIN-1-YL)ACETYL]-2-PROPOXYPHENYL}-6-(PROPAN-2-YL)PYRIMIDIN-4(3H)-ONE MG:MAGNESIUM ION PEG:DI(HYDROXYETHYL)ETHER ZN:ZINC ION | ||
4ia0 | [A] | [A] | [A] | 2.17 | 5BB:5-BROMO-2-{2-ETHOXY-5-[(4-METHYLPIPERAZIN-1-YL)SULFONYL]PHENYL}-6-OCTYLPYRIMIDIN-4(3H)-ONE MG:MAGNESIUM ION ZN:ZINC ION | ||
4myq | [A] | [A] | [A] | 1.9 | 19T:(4-{[2-(5-CHLOROTHIOPHEN-2-YL)-5-ETHYL-6-METHYLPYRIMIDIN-4-YL]AMINO}PHENYL)ACETIC ACID EDO:1,2-ETHANEDIOL MG:MAGNESIUM ION NA:SODIUM ION ZN:ZINC ION | ||
4npv | [A] | [A] | [A] | 2.4 | 0NK:6,7,8-TRIMETHOXY-N-(PENTAN-3-YL)QUINAZOLIN-4-AMINE MG:MAGNESIUM ION ZN:ZINC ION | ||
4npw | [A] | [A] | [A] | 1.9 | 0NY:7,8-DIMETHOXY-N-[(2S)-1-(3-METHYL-1H-PYRAZOL-5-YL)PROPAN-2-YL]QUINAZOLIN-4-AMINE MG:MAGNESIUM ION ZN:ZINC ION | ||
4nw7 | [A] | [A] | [A] | 2.15 | 2O5:(4-{[4-(3-CHLOROPHENYL)-6-CYCLOPROPYL-1,3,5-TRIAZIN-2-YL]AMINO}PHENYL)ACETIC ACID EDO:1,2-ETHANEDIOL MG:MAGNESIUM ION NA:SODIUM ION ZN:ZINC ION | ||
4oew | [A] | [A] | [A] | 2.44 | 5IO:6-ETHYL-5-IODO-2-{5-[(4-METHYLPIPERAZIN-1-YL)SULFONYL]-2-PROPOXYPHENYL}PYRIMIDIN-4(3H)-ONE MG:MAGNESIUM ION ZN:ZINC ION | ||
4oex | [A] | [A] | [A] | 2.14 | 5EO:6-ETHYL-2-{5-[(4-METHYLPIPERAZIN-1-YL)SULFONYL]-2-PROPOXYPHENYL}PYRIMIDIN-4(3H)-ONE MG:MAGNESIUM ION ZN:ZINC ION | ||
5b25 | [A] | [A] | [A] | 1.9 | 4QJ:(11R,15S)-4-{[4-(6-FLUOROPYRIDIN-2-YL)PHENYL]METHYL}-8-METHYL-5-(PHENYLAMINO)-1,3,4,8,10-PENTAAZATETRACYCLO[7.6.0.02,6.011,15]PENTADECA-2,5,9-TRIEN-7-ONE GOL:GLYCEROL MG:MAGNESIUM ION SO4:SULFATE ION ZN:ZINC ION | ||
5uoy | [A] | [A] | [A] | 1.82 | 8HM:6-[(4-METHOXYPHENYL)METHYL]-9-[(OXAN-4-YL)METHYL]-8,9,10,11-TETRAHYDROPYRIDO[4___sq___,3___sq___:4,5]THIENO[3,2-E][1,2,4]TRIAZOLO[1,5-C]PYRIMIDIN-5(6H)-ONE MG:MAGNESIUM ION ZN:ZINC ION | ||
5up0 | [A] | [A] | [A] | 2.04 | 8HP:6-[(4-CHLOROPHENYL)METHYL]-8,9,10,11-TETRAHYDRO[1]BENZOTHIENO[3,2-E][1,2,4]TRIAZOLO[1,5-C]PYRIMIDIN-5(6H)-ONE MG:MAGNESIUM ION ZN:ZINC ION | ||
5w6e | [A] | [A] | [A] | 1.9 | 0NY:7,8-DIMETHOXY-N-[(2S)-1-(3-METHYL-1H-PYRAZOL-5-YL)PROPAN-2-YL]QUINAZOLIN-4-AMINE MG:MAGNESIUM ION ZN:ZINC ION | ||
7lrc | [A2B2] | [A2B2] | [A2B2] | ELECTRON MICROSCOPY 2.97 |
MG:MAGNESIUM ION MN:MANGANESE (II) ION X5M:(4~{R})-3-[4-(DIETHYLAMINO)-3-[OXIDANYL(OXIDANYLIDENE)-$L^{4}-AZANYL]PHENYL]-4-METHYL-4,5-DIHYDRO-1~{H}-PYRIDAZIN-6-ONE |
*Chain Formula of OLIGAMI.
[ ] : Polypeptide - [AB] : Protein, [ab] : Small peptide
( ) : Nucleic acid - (AB) : DNA, (ab) : RNA
[ ] : Polypeptide - [AB] : Protein, [ab] : Small peptide
( ) : Nucleic acid - (AB) : DNA, (ab) : RNA